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. 2023 Feb;103(2):63–76. doi: 10.1124/molpharm.122.000591

TABLE 4.

α7-selective agonists

HS activation HS TQS LS activation LS TQS
4a. Responses Average ± S.D. Average ± S.D. Average ± S.D. Average ± S.D.
GTS-21 0.103 ± 0.023 34.514 ± 11.300 0.012 ± 0.004 0.753 ± 0.173
PNU-282987 0.014 ± 0.018 0.566 ± 0.298 0.009 ± 0.012 0.142 ± 0.147
TC-1698 0.013 ± 0.003 7.197 ± 1.694 0.009 ± 0.002 0.545 ± 0.199
AR-R17779 0.008 ± 0.006 3.017 ± 0.847 0.007 ± 0.007 0.109 ± 0.039
choline 0.022 ± 0.005 12.702 ± 6.048 0.024 ± 0.009 0.885 ± 0.237

See Supplemental Material for ANOVA results.