. 2023 Jan 4;66(2):1301–1320. doi: 10.1021/acs.jmedchem.2c01460

Table 3. Activity of C-3 Substituted Analogues^a^,^b.

graphic file with name jm2c01460_0011.jpg

IC₅₀ (pIC₅₀ ± SEM) values (μM) and PDB IDs are reported.

>Denotes less than 50% inhibition in the reported highest concentration, and ≫ denotes no inhibition at the reported concentration; *value limited by the protein concentration used.

Table 3. Activity of C-3 Substituted Analoguesa,b.

Table 3. Activity of C-3 Substituted Analogues^a^,^b.