Table 7.

Synthesis of 1-Phenylcyclopropane carboxamide derivatives (8a–8t).

S.No	Acid	Amine	Product	Yield (%)
1	3a	7	8a	85
2	3a	5a	8b	72
3	3a	5b	8c	84
4	3a	5c	8d	81
5	3b	7	8e	78
6	3b	5a	8f	76
7	3b	5b	8g	81
8	3c	7	8h	83
9	3c	5a	8i	76
10	3d	5a	8j	79
11	3d	5b	8k	71
12	3e	7	8l	79
13	3e	5a	8m	84
14	3e	5b	8n	88
15	3e	5c	8o	91
16	3f	7	8p	72
17	3f	5a	8q	80
18	3f	5b	8r	83
19	3g	5a	8s	73
20	3g	5b	8t	88

*All reactions were carried out on a 10 mg scale. The reaction was monitored by TLC and LCMS. Acid (1.0 eq), Amine (1.0 eq), HATU (1.5 eq), DIPEA (3.0 eq), DMF (5 vol).