Table 2.
Effect of some parameters (solvent and amount of catalyst) for the preparation of 4a.
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|---|---|---|---|---|---|
| Entry | Catalyst (mg) | Solvent | Temperature (°C) | Time (min) | Yield (%) |
| 1 | Fe3O4@CPTMO-phenylalanine-Ni (0) | Water | Reflux | 720 | 0 |
| 2 | Fe3O4@CPTMO-phenylalanine-Ni (30) | Water | Reflux | 25 | 85 |
| 3 | Fe3O4@CPTMO-phenylalanine-Ni (30) | Acetone | Reflux | 30 | 80 |
| 4 | Fe3O4@CPTMO-phenylalanine-Ni (20) | Water/Acetone (2:1) | 80 | 30 | 88 |
| 5 | Fe3O4@CPTMO-phenylalanine-Ni (30) | Water/Acetone (2:1) | 80 | 3 | 98 |
| 6 | Fe3O4@CPTMO-phenylalanine-Ni(30) | Ethanol | Reflux | 45 | 70 |
| 7 | Fe3O4@CPTMO-phenylalanine-Ni (30) | n-Hexane | Reflux | 60 | 43 |
| 8 | Fe3O4@CPTMO-phenylalanine-Ni (40) | Water/Acetone (2:1) | 80 | 30 | 90 |
| 9 | Fe3O4 (30) | Water/Acetone (2:1) | 80 | 300 | 68 |
| 10 | Fe3O4@CPTMO (30) | Water/Acetone (2:1) | 80 | 250 | 78 |
| 11 | Fe3O4@CPTMO-phenylalanine (30) | Water/Acetone (2:1) | 80 | 180 | 82 |
