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Primary in vitro pharmacokinetic (PK) data for 24
| Parameter | Value |
|---|---|
| Kinetic solubility [×10−6 m] | 47.2 |
| Calu‐3 (Papp) [10–6 cm s−1] | 3.1 ± 0.28 |
| Mouse liver S9 t½ [min] | 50 |
| Mouse hepatocytes t½ [min] | 9 |
| Plasma binding human [%] | >99 |
| Plasma binding murine [%] | >99 |
