TABLE 2.
Selected 6A1HI analogues from SAR studies
Compound | Structure | DENV-R2A replication (fold DMSO) | Cell viability (fold DMSO) |
---|---|---|---|
6A1HI |
![]() |
0.04 | 0.93 |
3 |
![]() |
1.10 | 0.93 |
7 |
![]() |
1.05 | 1.07 |
18 |
![]() |
1.06 | 0.98 |
6 |
![]() |
0.96 | 0.76 |
75 |
![]() |
1.06 | 0.99 |
9 |
![]() |
0.90 | 1.03 |
52 |
![]() |
1.15 | 0.93 |
76 |
![]() |
0.87 | 0.98 |
4 |
![]() |
0.97 | 0.75 |
42 |
![]() |
1.07 | 0.93 |