Table V.
Oral Dosage, Onset Time, Duration of Effects and Half-life of Selected DBZDs (59–62)
Compound | “Recreational” oral doses [mg] | Onset [min] | Duration of effects [h] | Half- life [h] |
---|---|---|---|---|
3-Hydroxyphenazepam | 0.5–4 | 30–90 | 24 | N/A |
Clonazolam | 0.2–1 | 20–60 | 6–10 | 3.6 |
Deschloroetizolam | 4–6 | 1–5 | 8–10 | N/A |
Diclazepam | 2–4 | 15–90 | 8–12 | 42 |
Etizolam | 0.25–3 Therapeutic: 0.5–2.0 |
30–120 | 5–8 | 3.4–7.1 |
Flualprazolam | 0.125–2.5 | 10–30 | 6–14 | 9.5–12 |
Flubromazepam | 4–8 | 15–90 | 12–18 | 106 |
Flubromazolam | 0.15–0.25 | 20–45 | Sedation for 10 h, Partial amnesia >24 h |
Possibly 30 h |
Flunitrazolam | 0.08–0.15 | 10–30 | 4–5 | N/A |
Meclonazepam | 2–3 | 20–60 | 9–15 | 80 |
Metizolam | 2 | 30–90 | 5–8 | N/A |
Nifoxipam | 0.5–3.0 | 45–120 | 10–75 | N/A |
Norflurazepam (N-desalkylflurazepam) |
5–10 | 45–120 | 10–16 | 40–250 |
Phenazepam | 3–5 Therapeutic: max. 10 |
15–60 | >18 | 15–60 |
Pyrazolam | 0.5–4 | 10–25 | 5–8 | 17 |