Table 7.
Pharmacokinetics of G1 in rats following intravenous and oral administration (n = 3).
| Parameter | G1 (n = 3) |
G1 (n = 3) |
|---|---|---|
| iv (10 mg / kg) | po (50 mg / kg) | |
| Tmax(h) | 0.03 | 0.25 |
| Cmax(nM) | 3.77 | 2.92 |
| t1/2(h) | 5.72 | 5.55 |
| CL(L / h / kg) | 0.29 | 1.70 |
| VZ(L / kg) | 2.39 | 13.12 |
| AUC(0–8) (nM∙h) | 6.13 | 6.39 |
| AUC(0−∞) (nM∙h) | 11.47 | 10.15 |
| F (%) | 20.85 |