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. 2009 Jan 15;9:e6.

Table 3.

Medications implicated in gynecomastia3,5,11

Hormones
   Estrogens and estrogen agonists
   Androgens and anabolic steroids
   Human chorionic gonadotropin
Androgen antagonists
   Ketoconazole
   Flutamide
   Metronidazole
   Finasteride
   Spironolactone
   Etomidate
Antiulcer drugs
   Cimetidine
   Omeprazole
   Ranitidine
Cytotoxic agents
   Bisulfar
   Vincristine
   Nitrosoureas
   Procarbazine
   Cisplatin
   Methotrexate
   Cyclophosphamide
   Chlorambucil
Psychoactive drugs
   Tricyclic antidepressants
   Phenothiazines
   Diazepam
Cardiovascular agents
   Amiodarone
   Angiotensin-converting enzyme inhibitors
   Calcium channel blockers
   Digitoxin
   Methyldopa
Antituberculotic agents
   Ethionamide
   Thiacetazone
   Isoniazid
Antiviral therapeutics
   Protease inhibiters
Miscellaneous
   Marijuana
   Heroine
   Methadone
   Alcohol
   Amphetamines
   Phenytoin
   Penicillamine