Table 2. Summary of brain and spinal cord exposure of 8D3130, 8D3130-PMO, and NIP228 in C57BL/6J mice following intravenous administration.
Construct | Brain | Spinal cord | ||||
---|---|---|---|---|---|---|
Tmax (h) | Cmax (μg/g) | AUClast (h×μg/g) | Tmax (h) | Cmax (μg/g) | AUClast (h×μg/g) | |
8D3130 | 24 | 22.6 | 2,180 | 24 | 12.6 | 1,460 |
8D3130-PMO | 24 | 13 | 1,330 | 24 | 10.5 | 614 |
NIP228 | 24 | 2.29 | 263 | 24 | 1.79 | 28.4 |
Tmax, time to maximum concentration.