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. Author manuscript; available in PMC: 2019 Feb 19.
Published in final edited form as: Bioorg Med Chem. 2018 Mar 19;26(11):2984–2991. doi: 10.1016/j.bmc.2018.03.030

Figure 4.

Figure 4

AlphaScreen binding assay for H3K4me3 and His-KDM7(PHD). Normalised dose-response inhibition curves for the displacement of H3K4me3-Bn from KDM7A/B/C by representative AMI derivatives.