Table 1: Ribociclib pharmacokinetic parameters summary in mice bearing mouse tumor #2416 (n=7).
AUC-0–24h, Area under concentration-time curve from time zero to 24 h after dose; tECF, tumor extracellular fluid.
Parameters [Unit] | Mean Estimates (SD) |
---|---|
Half-life [h] | 4.26 (0.737) |
Unbound Plasma AUC0–24h [ng × h/mL] | 5820 (926) |
tECF AUC0–24h/unbound Plasma AUC0–24h | 0.162 (0.119) |