Scheme 1.
Syntheses of the cpAbs a
aReagents and Conditions: (a) S21, THPTA, CuSO4, sodium ascorbate, H2O, t-BuOH, rt, 2 h, 4 100%, 5 67%; (b) mouse mAb 38C2, 100 mM PBS solution (pH 7.4), rt, 2 h.
Syntheses of the cpAbs a
aReagents and Conditions: (a) S21, THPTA, CuSO4, sodium ascorbate, H2O, t-BuOH, rt, 2 h, 4 100%, 5 67%; (b) mouse mAb 38C2, 100 mM PBS solution (pH 7.4), rt, 2 h.