Table 1.
| |||
---|---|---|---|
Entry | Ligand | Major Product, yieldc | Minor Product(s), yieldd |
1 |
3a 19%, 33% ee |
||
2 | |||
3b |
3a and 4a not observed |
Reaction conditions: [(coe)2RhCl]2 5 mol%, ligand 10 mol%, AgBF4 10 mol%, DCE (0.2 M), 40 °C, 36 h,
[(coe)2RhCl]2 2.5 mol%, ligand 5 mol%, AgBF4 5 mol%, 40 °C, 4 h,
Isolated yield,
Determined by GC-FID.
>20:1 dr, determined by 1H NMR.
one equivalent of 1a was used as a CO donor. DTBM: 3,5-di(tert-butyl)-4-methoxyphenyl