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. Author manuscript; available in PMC: 2018 Feb 20.
Published in final edited form as: Chem Rev. 2017 Mar 24;118(3):989–1068. doi: 10.1021/acs.chemrev.6b00801

Table 1.

Summary Table of Kinact/KI Data of LSD1 Inhibitorsa

inhibitor Kinact/KI (M−1 s−1) Ki (µM)
NCL-1 2000 ± 670 5.7 ± 2.4
S2101 4560 0.61
25 N.R. 1.3
RN-1 N.R. N.R.
26 4100 ± 980 0.75 ± 0.5
GSK2879552 1078 N.R.
27 1458 2.4
a

N.R. = not reported.