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. Author manuscript; available in PMC: 2018 Jun 26.
Published in final edited form as: Molecules. 2018 May 19;23(5):E1221. doi: 10.3390/molecules23051221

Table 2.

CaMKK2 FRET results for advanced TDZ analogues.

graphic file with name nihms971521u2.jpg
Compound R1 FRET (IC50) a Compound R1 FRET (IC50) a
1 graphic file with name nihms971521t8.jpg >50 14 graphic file with name nihms971521t9.jpg >50
2 graphic file with name nihms971521t10.jpg >50 15 graphic file with name nihms971521t11.jpg >50
3 graphic file with name nihms971521t12.jpg 34 16 graphic file with name nihms971521t13.jpg >50
10 graphic file with name nihms971521t14.jpg 7.8 17 graphic file with name nihms971521t15.jpg >50
11 graphic file with name nihms971521t16.jpg 3.2 18 graphic file with name nihms971521t17.jpg >50
12 graphic file with name nihms971521t18.jpg 10.5 19 graphic file with name nihms971521t19.jpg 38
13 graphic file with name nihms971521t20.jpg 43 - Ponatinib Staurosporine 0.4 & 0.0023
a

Average of 2 experiments for CaMKK2/(μM).