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. 1951 Nov 20;35(2):203–225. doi: 10.1085/jgp.35.2.203

ON THE EFFECT OF COCAINE UPON SODIUM-DEFICIENT FROG NERVE

R Lorente de Nó 1
PMCID: PMC2147291  PMID: 19873523

Abstract

Cocaine diffuses through the epineurium with remarkable rapidity. The coefficient of diffusion of cocaine in the epineurium cannot be less than 0.44 x 10–4 cm.2/min.; it probably is not less than 1.22 x 10–4 cm.2/min. Lack of sodium markedly sensitizes the nerve fibers to the anesthetic action of cocaine. With sodium-deficient A fibers the action of cocaine develops in two phases. During the first phase cocaine substitutes for sodium and restores to A fibers the ability to conduct impulses; during the second phase cocaine produces anesthesia. It is suggested that cocaine anesthetizes the nerve fibers through the sodium mechanism; i.e., by interfering with some of those chemical reactions in which, directly or indirectly, the internal sodium takes part.

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Selected References

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  1. FENG T. P., LIU Y. M. The connective tissue sheath of the nerve as effective diffusion barrier. J Cell Physiol. 1949 Aug;34(1):1–16. doi: 10.1002/jcp.1030340102. [DOI] [PubMed] [Google Scholar]
  2. LORENTE de NO R. The ineffectiveness of the connective tissue sheath of nerve as a diffusion barrier. J Cell Physiol. 1950 Apr;35(2):195–240. doi: 10.1002/jcp.1030350204. [DOI] [PubMed] [Google Scholar]
  3. LORENTE DE NO R. Equilibria of frog nerve with different external concentrations of sodium ions. J Gen Physiol. 1951 Sep;35(1):145–182. doi: 10.1085/jgp.35.1.145. [DOI] [PMC free article] [PubMed] [Google Scholar]

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