Table 1.
Relative kcat/Km | ||||
---|---|---|---|---|
Peptide | SIRT1 | SIRT2 | ySir2 | TbSir2 |
AcGG(AcK)AP | 1.7 ± 0.5 | 0.6 ± 0.1 | 1.5 ± 0.7 | 1.3 ± 0.2 |
AcTGG(AcK)AP | 0.5 ± 0.1 | 0.6 ± 0.1 | 1.6 ± 0.6 | 0.7 ± 0.2 |
AcSTGG(AcK)AP | 1.6 ± 0.5 | 0.8 ± 0.1 | 1.8 ± 0.8 | 0.6 ± 0.1 |
AcGG(AcK)APR | 0.7 ± 0.1 | 0.6 ± 0.1 | 2.5 ± 1.3 | 1.2 ± 0.2 |
AcTGG(AcK)APR | 0.6 ± 0.1 | 0.7 ± 0.1 | 1.7 ± 0.8 | 0.9 ± 0.2 |
AcSTGG(AcK)APR | 0.7 ± 0.1 | 0.9 ± 0.2 | 1.6 ± 0.8 | 1.4 ± 0.2 |
AcGG(AcK)APRK | 1.0 ± 0.2 | 0.7 ± 0.1 | 2.3 ± 0.9 | 1.8 ± 0.2 |
AcGG(AcK)APRKQ | 0.8 ± 0.2 | 0.7 ± 0.1 | 2.1 ± 0.8 | 1.4 ± 0.2 |
AcKSTGG(AcK)AP | 0.7 ± 0.1 | 0.6 ± 0.1 | 2.1 ± 0.8 | 1.8 ± 0.7 |
AcTGG(AcK)APRK | 1.0 ± 0.1 | 1.0 ± 0.1 | 1.0 ± 0.4 | 1.0 ± 0.1 |