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British Journal of Pharmacology logoLink to British Journal of Pharmacology
. 2009 Nov;158(Suppl 1):S241–S254. doi: 10.1111/j.1476-5381.2009.00507.x

Suppliers' Contact Details

PMCID: PMC2884678

A.G. Scientific Inc.

6450 Lusk Blvd. Suite E102

San Diego

CA 92121

USA

http://www.agscientific.com/

Alexis Biochemicals

AXXORA LLC

6181 Cornerstone Court East

Suite 103

San Diego

CA 92121

USA

http://www.Alexis-biochemicals.com/

Avanti Polar Lipids Inc.

700 Industrial Park Drive

Alabaster

AL 35007

USA

http://www.avantilipids.com

Bachem Bioscience Inc.

3700 Horizon Drive

King of Prussia

PA 19406

USA

http://www.bachem.com

BIOTREND Chemikalien GmbH

Eupener Str. 157

D-50933 Cologne

Germany

http://www.biotrend.com/

Calbiochem/EMD Biosciences

10394 Pacific Center Court

San Diego

CA 92121

USA

http://www.calbiochem.com

Sigma-Aldrich

PO Box 14508

Pollards Wood

St Louis

MO 63178-9916

USA

http://www.sigma-aldrich.com

Tocris Bioscience

Tocris House

Hung Road

Bristol

BS11 9XJ

UK

http://www.tocris.com

Amersham Biosciences UK Ltd

GE Healthcare

Nightingales Lane

Chalfont St Giles

Buckinghamshire HP8 4SP

UK

http://www.amershambiosciences.com

A. Menarini Pharma UK SRL

Menarini House

Mercury Park

Wycombe Lane

Wooburn Green

High Wycombe

Buckinghamshire HP10 OHH

UK

http://www.menarini.com

Roche Pharmaceuticals

Pharmaceuticals Division

Grenzacherstrasse 124

CH-4070 Basel

Switzerland

http://www.roche.com

Compound Name Compound Supplier
(−)-(S)-BAYK8664 (−)-(S)-methyl-1,4-dihydro-2,6-dimethyl-3-nitro-4-(2-trifluromethylphenyl)-pyridine-5-carboxylate Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
(+)7-OH-DPAT (+)-7-hydroxy-2-aminopropylaminotetralin Sigma-Aldrich, Tocris Bioscience
(+)-Tc (+)-Tubocurarine Alexis Biochemicals, BIOTREND, Sigma-Aldrich
(RS)PPG (R,S)-4-phosphonophenylglycine Alexis Biochemicals, BIOTREND, Tocris Bioscience
(S)-3, 4-DCPG (S)-3,4-dicarboxylphenylglycine BIOTREND, Tocris Bioscience
[Ala1, 3, 11, 15]ET-1 Alexis Biochemicals, Bachem, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
[Ala11, d-Leu15]orexin-B Bachem, BIOTREND, Calbiochem, Tocris Bioscience
12-(S)-HPETE 12-(S)-hydroperoxyeicosatetraenoic acid BIOTREND
1400W N-(3-(aminomethyl)benzyl)acetamidine Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
15-(S)-HPETE 15-(S)-hydroperoxyeicosatetraenoic acid BIOTREND, Sigma-Aldrich
15deoxy-PGJ2 also known as 15-deoxy-Δ-12,14-PGJ2 BIOTREND, Sigma-Aldrich, Tocris Bioscience
1S, 3R-ACPD 1-aminocyclopentane-1S,3R-dicarboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
2-APB 2-amino ethoxyphenylborate BIOTREND, Calbiochem, Tocris Bioscience, Sigma-Aldrich
2Cl-IB-MECA 2-chloro-N6-(3-iodobenzyl)adenosine-5′-N-methyluronamide Sigma-Aldrich, Tocris Bioscience
2-MeSADP 2-methylthio-adenosine-5′-diphosphate BIOTREND, Sigma-Aldrich, Tocris Bioscience
2-MeSATP 2-methylthio-adenosine-5′-triphosphate BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
2R, 4R-APDC Aminopyrrolidine-2R,4R-dicarboxylate also known as LY314593 Alexis Biochemicals, BIOTREND, Tocris Bioscience
3-APMPA 3-amino-propyl-(p-methyl)-phosphinic acid, also known as CGP35024 Sigma-Aldrich, Tocris Bioscience
3-APPA (CGP27492) 3-amino-propyl-phosphinic acid
3HPG 3-hydroxyphenylglycine Sigma-Aldrich, Tocris Bioscience
4-AP 4-aminopyridine BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
4CPG 4-carboxyphenylglycine BIOTREND, Sigma-Aldrich, Tocris Bioscience
4-DAMP 4-diphenylacetoxy-N-methylpiperidine methiodide BIOTREND, Sigma-Aldrich, Tocris Bioscience
4P-PDOT 4-phenyl-2-propionamidotetraline BIOTREND, Tocris Bioscience
4a-PDD 4a-phorbol 12,13-didecanoate Alexis Biochemicals, BIOTREND, Calbiochem
5(S)-HETE 5(s)-hydroxy-6E,8z,11z,14z-eicosatetraenoic acid BIOTREND, Sigma-Aldrich
5-(S)-HETE 5-(S)-hydroeicosatetraenoic acid Sigma-Aldrich
5(S)-HpETE 5(s)-hydroperoxy-6E,8z,11z,14z-eicosatetraenoic acid BIOTREND
5-CT 5-carboxamidotryptamine BIOTREND, Sigma-Aldrich, Tocris Bioscience
5-fluoro-20-deoxyuridine BIOTREND, Calbiochem, Sigma-Aldrich
5-fluorouridine Sigma-Aldrich
5MCA-NAT 5-methoxy-carbonylamino-N-acetyltryptamine, also known as GR 135531 BIOTREND, Sigma-Aldrich, Tocris Bioscience
5-oxo-ETE 5-oxo-6E,8z,11z,14z-eicosatetraenoic acid
6-iodo-nor dihydrocapsaicin also known as 6-iodonor dihydrocapsaicin BIOTREND, Tocris Bioscience
7NI 7-nitroindazole Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
8-OH-DPAT 8-hydroxy-2-(di-n-propylamino)tetralin BIOTREND, Sigma-Aldrich, Tocris Bioscience
9-AC Anthracene-9-carboxylic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
A61603 N-(5-[4,5-dihydro-1H-imidazol-2-y]-2-hydroxy-5,6,7,8-tetrahydronaphthalen-1-yl) methanesulphonamide hydrobromide BIOTREND, Tocris Bioscience
AB-MECA N6-(4-aminobenzyl)-adenosine-5′-N-methyluronamide BIOTREND, Sigma-Aldrich
ABT229 8,9-anhydro-4″-deoxy-3′-N-desmethyl-3′-N-ethylerythromycin B 6, 9-hemiacetal
ABT-418 (S)-3-methyl-5-(1-methyl-2-pyrrolidinyl) isoxazole Sigma-Aldrich
AC187 acetyl-[Asn30,Tyr32]salmon calcitonin Bachem, Calbiochem, Sigma-Aldrich
ACh Acetylcholine BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
A-conotoxin-GIC Calbiochem
Adenophostin A Calbiochem
AFDX384 (±)-5,11-dihydro-11-([{2-(2-N,N-[dipropylamino]methyl)piperidin-1-yl} BIOTREND, Tocris Bioscience
ethylamino]carbonyl)-6H-pyrido[2,3-b](1,4)benzodiazepine-6-one
AG-3-5 1-[2-hydroxyphenyl]-4[3-nitrophenyl]-1,2,3,6-tetrahydropyrimidine-2-one BIOTREND, Sigma-Aldrich, Tocris Bioscience
AGN192093 (Z)-7-([1a,5a,6a,7b]-7-[{1E,3S}-3-hydroxy-1-octenyl]-3-oxo-2,4-dioxobicyclo[3.2.1]oct-6-yl)-5-heptenol Sigma-Aldrich
AH13205 trans-2-(4-[1-hydroxyhexyl]phenyl)-5-oxocyclopentaneheptanoate Sigma-Aldrich
AH23848 (1a[z],2b,5a)-(7)-7-(5-[{(1,1′-biphenyl)-4-yl}methoxy]-2-[4-morpholinyl]-3-oxocyclopentyl)-4-heptenoate Sigma-Aldrich
AIDA 1-aminoindan-1,5(RS)-dicarboxylic acid, also known as UPF523 Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
AM1241 (2-iodo-5-nitro-phenyl)-[1-(1-methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-methanone Alexis Biochemicals, Sigma-Aldrich
AM251 N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
AM281 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carboxamide Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
AM630 6-iodopravadoline Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
AMA S-(5′-deoxy-5′-adenosyl)-methylthioethyl-hydroxylamine
AMPA (RS)-α-amino-3-hydroxy-5-methyl-4-isoxazole proprionic acid Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Ana-a Anatoxin-a BIOTREND, Tocris Bioscience
Anandamide Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris BiosciencE
Antalarmin N-butyl-N-ethyl-(2,5,6-trimethyl)-7-[2,4,6-trimethylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl-amine Sigma-Aldrich, Tocris Bioscience
AOAA Aminooxyacetic acid Bachem
APA 1-aminooxy-3-aminopropane
Apamin Alexis Biochemicals, Bachem, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
APTA (RS)-2-amino-3-(3-hydroxy-5-tert-butylisoxazol-4-yl)propionic acid
ARC239 2-[2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl]-4,4-dimethyl-1,3-(2H,4H)-isoquinolindione dihydrochloride BIOTREND, Tocris Bioscience
ARF ADP-ribosylation factor Calbiochem
Astemizole BIOTREND, Sigma-Aldrich
Astressin cyc 30–33[d-Phe12,Nle21,38,Glu30,Lys33]CRF-(12-41) Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
ATPO (RS)-2-amino-3-(3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid Sigma-Aldrich
ATPγS Adenosine 5′-(3-thio)triphosphate Alexis Biochemicals, Calbiochem, Roche, Sigma-Aldrich
atr Atropine BIOTREND, Calbiochem, Sigma-Aldrich
ATRA All-trans-retinoic acid BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Azelaoyl-PAF 1-O-hexadecyl-2-O-(9-carboxyoctanoyl)-sn-glyceryl-3-phosphocholine Alexis Biochemicals, Avanti, Sigma-Aldrich
AZT 3′-azido-3′-deoxythymidine Calbiochem, Sigma-Aldrich
B9958 Lys-Lys[Hyp3,Cpg5,dTic7,Cpg8][des-Arg9]BK
BADGE bisphenol A diglycidyl ether Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
BAYu9773 6(R)-(4′-carboxyphenyl-thio)-5(S)-hydroxy-7(E),11(Z),14(Z)-eicosatetraenoic acid BIOTREND, Sigma-Aldrich
BDS-1 blood depressing substance Calbiochem
Bezafibrate 2-[4-[2-(4-Chlorobenzamido)ethyl]phenoxy]-2-methylpropanoic acid BIOTREND, Calbiochem, Sigma-Aldrich
Bgt α-Bungarotoxin Alexis BiochemicalsBIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
BHT920 6-allyl-2-amino-5,6,7,8-tetrahydro-4H-thiazolo-[4,5-d]-azepine Sigma-Aldrich, Tocris Bioscience
BIBP3226 R-N2-(diphenylacetyl)-N-(4-hydroxyphenyl)methyl-argininamide Bachem, Sigma-Aldrich, Tocris Bioscience
BIM23056 DPhe-Phe-Tyr-dTrp-Lys-Val-Phe-dNal-NH2 BIOTREND, Tocris Bioscience
BIM23127 d-Nal-cyc[Cys-Tyr-d-Trp-Orn-Val-Cys]-Nal-NH2 Bachem, BIOTREND, Tocris Bioscience
BMY45778 3-(4-[4,5-diphenyl-2-oxazolyl]-5-oxazolyl)phenoxyacetic acid BIOTREND, Tocris Bioscience
BMY7378 8-(2-[4-{2-methoxyphenyl}-1-piperazinyl]ethyl)-8-azaspiro[4,5]decane-7,9-dione dihydrochloride BIOTREND, Sigma-Aldrich, Tocris Bioscience
BN52021 (±)-trans-2,5-bis(3,4,5-trimethoxyphenyl)-1,3-dioxolane Sigma-Aldrich, Tocris Bioscience
bosentan
BQ123 cyc(dTrp-dAsp-Pro-dVal-Leu) Alexis Biochemicals, Bachem, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
BQ3020 N-acetyl-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp Alexis Biochemicals, Bachem, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
BQ788 N-cis-2,6-dimethylpiperidinocarbonyl-l-γ-methylleucyl-d-1-methoxycarboyl-d-norleucine Alexis Biochemicals, Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
BRL15572 3-[4-(3-chlorophenyl) piperazin-1-yl]-1,1,-diphenyl-2-propanol BIOTREND, Sigma-Aldrich, Tocris Bioscience
BRL37344 Sodium 4-(2-[2-hydroxy-3-chlorophenyl}ethylamino]propyl)phenoxyacetate Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
BRL44408 2-(2H-[1-methyl-1,3-dihydroisoindole]methyl)-4,5-dihydroimidazole BIOTREND, Sigma-Aldrich, Tocris Bioscience
BRL54443 3-(1-methylpiperidin-4-yl)1H-indol-5-ol BIOTREND, Sigma-Aldrich, Tocris Bioscience
BW245C 5-(6-carboxyhexyl)-1-(3-cyclohexyl-3-hydroxypropyl)hydantoin Sigma-Aldrich
BW723C86 1-[5(2-thienylmethoxy)-1H-3-indolyl]propan-2-amine hydrochloride Sigma-Aldrich, Tocris Bioscience
BWA868C 3-benzyl-5-(6-carboxyhexyl)-1-(2-cyclohexyl-2-hydroxyethylamino)hydantoin Sigma-Aldrich
C16:0 Palmitic acid BIOTREND, Calbiochem, Sigma-Aldrich
C18:0 Stearic acid BIOTREND, Calbiochem, Sigma-Aldrich
C18:1 Oleic acid BIOTREND, Calbiochem, Sigma-Aldrich
C18:2 Linoleic acid BIOTREND, Calbiochem, Sigma-Aldrich
C18:3, n-6 γ-linolenic acid BIOTREND
C2 Acetic acid Sigma-Aldrich
C20:4 Arachidonic acid BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
C20:5, n-3 Eicosapenta(5z,8z,11z,14z,17z)enoic acid BIOTREND
C22:6, n-3 Docosahexa(4z,7z,10z,13z,16z,19z)enoic acid
C3 Propionic acid Sigma-Aldrich
C4 Butyric acid Sigma-Aldrich
C7 Galanin-1–13-spantide Bachem, BIOTREND, Calbiochem, Sigma-Aldrich
Caffeine 1,3,7-trimethylxanthine Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Calciseptine BIOTREND
Calphostin C Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
CaM Calmodulin Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich
CCPA 2-chloro-N6-cyclopentyladenosine BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP12177A (−)-4-(3-tert-butylamino-2-hydroxypropoxy)-benzimidazol-2-one BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP20712A 2-hydroxy-5-(2-[{2-hydroxy-3-(4-[1-methyl-4-trifluoromethyl-2-imidazolyl]phenoxy propyl}amino]ethoxy)benzamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP35024 3-amino-propyl-(p-methyl)-phosphinic acid, also known as 3-APMPA Alexis Biochemicals
CGP35348 p-(3-aminopropyl)-p-diethoxymethylphosphinic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP37849 (RS)-(E)-2-amino-4-methylphosphono-3-pentanoic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP42112A Nicotinic acid-Tyr-(N-benzoylcarbonyl-Arg)-Lys-His-Pro-Ile-OH Bachem, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
CGP54626 [S-(R,R)]-[3-[[1-(3,4-dichlorophenyl)ethyl]amino]-2-hydroxypropyl](cyclohexylmethyl)phosphinic acid BIOTREND, Tocris Bioscience
CGP55845 3-[-1-(S)-(3,4-dichlorphenyl)-ethyl]amino-2(S)-hydroxypropyl-(p-benzyl)-phosphinic acid BIOTREND, Tocris Bioscience
CGP61594 (7)-trans-4-[2-(4-azidophenyl)acetylamino]-5,7-dichloro-1,2,3,4-tetrahydroquinoline-2-carboxylic acid
CGP62349 [3-[1-R-[[3-(methoxyphenylmethyl)hydroxyphosphinyl]-2(5)-hydroxypropyl]amino]ethyl]-benzoic acid
CGP64213 [3-[-(R)-[[3-5N-[1-[2-[[3-iodo-4-hydroxyphenyl]ethyl]carboxamido]pentyl]hydroxyphosphinyl]-2(S)-hydroxy-propyl]amino]ethyl-benzoic acid
CGP71683A Trans-naphthalene-1-sulphonic acid(4-[4-amino-quinazolin-2-ylamino]-methyl)-cyclohexylmethyl-amide hydrochloride BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGP7930 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGS15943 5-amino-9-chloro-2-(2-furyl)1,2,4-triazolo[1,5-c]quinazoline BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGS19755 4-phosphonomethyl-2-piperidinecarboxylic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGS21680 2-(4-[2-carboxyethyl]-phenethylamino)adenosine-5′-N-ethyluronamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
CGS25019C 4-(5-[4-{aminoiminomethyl}phenoxy]pentoxy)-3-methoxy-N,N-bis(1-methylethyl)benzamide-(Z)-2-butenedioate
Charybdotoxin Alexis Biochemicals Biochemicals, Bachem, BIOTREND, Calbiochem,
Aldrich, Tocris Bioscience
Chelerythrine Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
cho Choline Sigma-Aldrich
CHPG (RS)-2-chloro-5-hydroxyphenylglycine BIOTREND, Tocris Bioscience
CI966 (1-[2-{bis-4(trifluromethyl)phenyl}methoxy]ethyl)-1,2,5,6-tetrahydro-3-pyridinecarboxylic acid BIOTREND, Tocris Bioscience
CI977 (5R)-(5α,7α,8β)-(–)-N-methyl-N-(7-[1-pyrrolidinyl]-1-oxaspiro[4,5]dec-8-yl)-4-benzofuranacetamide monohydrochloride
Ciglitizone (±)-5-[4-(1-Methylcyclohexylmethoxy)benzyl]thiazolidine-2,4-dione Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Biochemicals
CJ13610 1-carboxamido-1-(3-S-[4-{2-methylimididazole}-thiophenyl])-4-cyclopentylether
CL316243 Disodium (R,R)-5-(2-[{2-(3-chlorophenyl)-2-hydroxyethyl}-amino]propyl)-1,3-benzodioxole-2,2,dicarboxylate BIOTREND, Tocris Bioscience
Clofibrate Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Biochemicals
CNQX 6-cyano-7-nitroquinoxaline-2,3-dione Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
CP101606 (1S,2S)-1-4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidino)-1-propanol
CP105696 (+)-1-(3S,4R)-[3-(4-phenylbenzyl)-4-hydroxy-chroman-7-yl]cyclopentane carboxylic acid
CP195543 (+)-2-(3-benzyl-4-hydroxychroman-7-yl)-4-trifluoromethylbenzoic acid
CP55940 (−)-3-[2-hydroxy-4-(1,1-dimethylheptyl)phenyl]-4-(3-hydroxypropyl)cyclohexan-1-ol BIOTREND, Sigma-Aldrich, Tocris Bioscience
CPA N6-cyclopentyladenosine BIOTREND, Sigma-Aldrich, Tocris Bioscience
CPCCOEt cyclopropan[b]chromen-1a-carboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
CpG DNA enriched in cytosine:guanosine pairs
CPP (±)-2-carboxypiperazine-4-yl)propyl-1-phosphonic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
CTOP DPhe-Cys-Tyr-dTrp-Lys-Thr-Pen-The-NH2 BIOTREND, Sigma-Aldrich, Tocris Bioscience
Cyt Cytosine Sigma-Aldrich
DAMGO Tyr-dAla-Gly-[NMePhe]-NH(CH2)2 Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
D-AP5 D(2)-2-amino-5-phosphonopentanoate BIOTREND, Sigma-Aldrich, Tocris Bioscience
dBzATP 2′,3′-O-di(benzoyl)-adenosine triphosphate
DCG-IV (2S,1′R,2′R,3′R)-2-(2,3-dicarboxycyclopropyl)glycine BIOTREND, Tocris Bioscience
DCKA dichlorokynurenic acid Alexis Biochemicals, Sigma-Aldrich, Tocris Bioscience
DCPIB 4-(2-butyl-6,7-dichlor-2-cyclopentyl-indan-1-on-5-yl) oxybutyric acid Tocris Bioscience
DD161515 N-[2-(2-(N-methylpyrrolidinyl)ethyl)glycyl]-[N-[2,4-dichlorophenethyl]glycyl]-N-(2,4-dichlorophenethyl)glycinamide Sigma Aldrich
DFMO α-difluoromethyl-l-ornithine, also known as eflornithine; Bachem, Calbiochem, Sigma-Aldrich, Tocris Bioscience
DGPP 8:0 dioctanoylglycerol pyrophosphate Avanti
DH97 2-benzyl-N-pentanoyltryptamine BIOTREND, Tocris Bioscience
DHA 4z,7z,10z,13z,16z,19z-docosahexaenoic acid Sigma-Aldrich
DHPG S-3,5-dihydroxyphenylglycine BIOTREND, Sigma-Aldrich, Tocris Bioscience
DHβE dihydro-β-erythroidine BIOTREND, Tocris Bioscience
Diazoxide 7-Chloro-3-methyl-2H-1,2,4-benzothiadiazine 1,1-dioxide BIOTREND, Sigma-Aldrich, Tocris Bioscience
diBA-(5)-C4 Bis-(1,3-dibutylbarbituric acid)pentamethine oxanol Sigma-Aldrich
Didanosine Sigma-Aldrich
BDIDS 4,4′-diisothiocyanostilbene-2,2′-disulphonic acid Calbiochem, Sigma-Aldrich
Diltiazem (2S,3S)-(+)-cis-3-Acetoxy-5-(2-dimethylaminoethyl)-2,3-dihydro-2-(4-methoxyphenyl)-1,5-benzothiazepin-4(5H)-one BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
dl-TBOA dl-threo-β-benzyloxyaspartate Tocris Bioscience
DMAB 3-(4)-dimethylaminobenzylidine anabaseine Tocris Bioscience
DMAC 3-(4)-dimethylaminocinnamylidine anabaseine
DMCM methyl-6,7-dimethoxy-4-ethyl-b-carboline-3-carboxylate BIOTREND, Sigma-Aldrich
DMPP 1,1-dimethyl-4-phenylpiperazinium BIOTREND, Sigma-Aldrich
DNQX 6,7-dinitroquinoxaline-2,3-dione Alexis Chemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
DOPA 3,4-dihydroxyphenylalanine Sigma-Aldrich
DPCPX 8-cyclopentyl-1,3-dipropylxanthine BIOTREND, Sigma-Aldrich, Tocris Bioscience
DPDPE cyc[dPen2,dPen5]enkephalin AG Scientific, Bachem, BIOTREND, Tocris Bioscience
d-Phe-CRF-(12-41) d-Phe12,Nle21,38,α MeLeu37-CRF Bachem, Tocris Bioscience
d-Trp8-g-MSH BIOTREND
ECDCA 6a-ethyl-chenodeoxycholate, also known as INT747
EF1502 N-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-hydroxy-4-(methylamino)4,5,6,7,tetrabenzo[d]isoxazol-3-ol
EGLU (S)-α-ethylglutamate Alexis Biochemicals, BIOTREND, Tocris Bioscience
EHNA erythro-9-(2-hydroxy-3-nonyl)adenine BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
EIPA ethylisopropylamiloride Sigma-Aldrich
EPA 5z,8z,11z,14z,17z-eicosapentaenoic acid or eicosapentaenoic acid BIOTREND, Calbiochem, Sigma-Aldrich
Epi epibatidine BIOTREND, Sigma-Aldrich, Tocris Bioscience
Erlotinib N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)quinazolin-4-amine, also known as OSI774 Sigma-Aldrich, Tocris Bioscience
exo-THPO 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazol
EXP3174 n-butyl-4-chloro-1-([2′-{1H-tetrazol-5yl}biphenyl-4-yl]methyl)imidazole-5-carboxylate
F180 Hmp-Phe-Ile-Hgn-Asn-Cys-Pro-Dab(Abu)-Gly-NH2
FAP10 Decanol phosphate
FAP12 Dodecanol phosphate
flAdipo full-length adiponectin
FMH α-Fluoromethylhistidine Sigma-Aldrich
Formycin B
FPL64176 2,5-dimethyl-4-[2(phenylmethyl)benzoyl]-H-pyrrole-3-carboxylate Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
FR139317 (R)2-([R-2-{(S)-2-([1-{hexahydro-1H-azepinyl}carbonyl]amino)methyl}pentanoyl]amino-3-(3-[methyl-1H-indodyl])propionylamino-3-(2-pyridyl))propionate Alexis Biochemicals, Tocris Bioscience
FR173657 (e)-3-(6-acetamido-3-pyridyl)-N-(N-[2,4-dichloro-3{(2-methyl-8-quinolinyl)oxymethyl}phenyl]-N-methylaminocarbonyl-methyl)acrylamide
gAdipo globular adiponectin Alexis Biochemicals, BIOTREND
GBR12935 1-(2-[diphenylmethoxy]ethyl)-4-(3-phenylpropyl)piperazine BIOTREND, Sigma-Aldrich, Tocris Bioscience
GC1 (3,5-dimethyl-4-[4-hydroxy-3-isopropylbenzyl]phenyloxy)acetate
GEA3162 1,2,3,4-oxatriazolium-5-amino-3-(3,4-dichlorophenyl)-chloride Alexis Biochemicals
gefitinib N-(3-chloro-4-fluoro-phenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine, also known as ZD1839
Gemcitabine
Ginkgolide B (±)-trans-2,5-bis(3,4,5-trimethoxyphenyl)-1,3-dioxolane; also known as (BN52021) BIOTREND, Sigma-Aldrich, Tocris Bioscience
Glibenclamide 5-Chloro-N-[2-[4-[[[(Cylcohexylamino)carbonyl]amino]sulphonyl]phenyl]ethyl]-2-methoxybenzamide Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
Go6983 Calbiochem, Sigma-Aldrich, Tocris Bioscience
GR100679 Cyclohexylcarbonyl-Gly-Ala-dTrp-Phe-NMe2
GR113808 [1-2[(methylsuphonyl)amino]ethyl]-4-piperidinyl]methyl-1-methyl-1H-indole-3-carboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
GR125743 n-[4-methoxy-3-(4-methyl-1-piperizinyl)phenyl]-3-methyl-4-(4-pyrindinyl)benzamide
GR159897 (R)-1-(2-[5-fluoro-1H-indol-3-yl]ethyl)-4-methoxy-4([phenylsulfinyl]methyl)piperidine BIOTREND, Sigma-Aldrich, Tocris Bioscience
GR32191 [1R-[1(Z),2b,3b,5]]-(+)-7-[5-[[(1,1′-biphenyl)-4-yl]methoxy]-3-hydroxy-2-(1-piperidinyl)cyclopentyl]-4-heptenoic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
GR55562 3-[3-(dimethylamino)propyl]-4-hydroxy-N-[4-(4-pyridinyl)phenyl]benzamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
GR64349 Lys-Asp-Ser-Phe-Val-Gly-(R-g-lactam) BIOTREND, Sigma-Aldrich, Tocris Bioscience
GR94800 N-α-benzoyl-Ala-Ala-dTrp-Phe-dPro-Pro-Nle-NH2 Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
GS39783 N,N′-dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine BIOTREND, Sigma-Aldrich, Tocris Bioscience
GTI 5-hydroxytryptamine-5-O-carboxymethylglycyltyrosinamide
GTS-21 3-(2,4)-dimethoxybenzylidine anabaseine (DMXB)
Guggulsterone trans-4,17(20)-pregnadiene-3,16-dione Sigma-Aldrich, Tocris Bioscience
GW273629 3-([2-{ethanimidoylamino}ethyl]sulphonyl)-l-alanine
GW274150 (S)-2-amino-(1-iminoethylamino)-5-thiopentanoic acid
GW3965 3-(3-[N-{2-chloro-3-trifluoromethylbenzyl}-{2,2-diphenylethyl}amino]propyloxy)phenylacetic acid hydrochloride Sigma-Aldrich, Tocris Bioscience
GW501516 2-methyl-4(((4-methyl-2-(4-trifluoromethylphenyl)-1,3-thiazol-5-yl)methyl)sulfanyl)phenoxy)acetic acid Sigma-Aldrich, Tocris Bioscience
GW583340 N-(3-chloro-4-[{3-fluorophenyl}-methoxy]-phenyl)-6-(2-[{(2-[methylsulfonyl]ethyl)amino}methyl]-4-thiazolyl)-4-quinazolinamine dihydrochloride
GW7647 2-([4-{2-([{cyclohexylamino}carbonyl][4-cyclohexylbutyl]amino)ethyl}phenyl]thio)-2-methylpropanoic acid BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
GW9662 2-chloro-5-nitro-N-phenylbenzamide Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
GYKI53655 1-(4-aminophenyl)-4-methyl-7,8-methylenedioxy-5H-(3N-methylcarbamate)-2,3-benzodiazepine; also known as HA966: 3-amino-1-hydroxypyrrolid-2-one Tocris Bioscience
HA966 3-amino-1-hydroxypyrrolid-2-one BIOTREND, Sigma-Aldrich, Tocris Bioscience
HC-3 hemicholinium-3 Sigma-Aldrich
HEAT 2-β-4-hydroxy-3-iodophenylethylaminomethyltetralone BIOTREND, Tocris Bioscience
HENECA 2-(1-(E)-hexenyl)adenosine-5′-N-ethyluronamide Sigma-Aldrich
hex hexamethenium
Himbacine (3S,3aR,4R,4aS,8aR,9aS)-4-[(1E)-2-[(2R,6S)-1,6-dimethyl-2-piperdinyl]ethenyl]decahydro-3- Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich
methylnaphtho[2,3-c]furan-1(3H)-one
HOE140 dArg[Hyp3,Thi5,dTic7,Oic8] bradykinin BIOTREND, Calbiochem,
HU308 {4-[4-(1,1-dimethylheptyl)-2,6-dimethoxy-phenyl]-6,6-dimethyl-bicyclo[3.1.1]hept-2-en-2-yl}-methanol
Iberiotoxin Alexis Biochemicals, Bachem, BIOTREND, Calbiochem, Sigma-
Aldrich, Tocris Bioscience
I-BOP (1S-[1α,2β{5Z},3α[1E,3S*],4α])-7-(3-[hydroxy-4-{4′-iodophenoxy}-1-butenyl]-7-oxabicyclo[2.2.1]hept-2-yl)-5-heptanoate
ICI118551 (−)-1-(2,3-[dihydro-7-methyl-1H-inden-4-yl]oxy)-3-([1-methylethyl]-amino)-2-butanol Sigma-Aldrich, Tocris Bioscience
IL-8 Interleukin 8 Bachem, BIOTREND, Calbiochem, Sigma-Aldrich
IP-10 γ-Interferon-inducible protein 10 Bachem, BIOTREND, Sigma-Aldrich
Ip5I Diinosine-5′,5″-pentaphosphate Calbiochem, Sigma-Aldrich
IRL1620 Suc[Glu9,Ala11,15]ET-1-(10–21) Alexis Biochemicals, Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
IRL2500 N-(3,5-dimethylbenzoyl)-N-methyl-(d)-(4-phenylphenyl)-Ala-Trp BIOTREND, Tocris Bioscience
BIvabradine (3-(3-{[((7S)-3,4-dimethoxybicyclo [4,2,0] octa-1,3,5-trien7-yl) methyl] methylamino}propyl)-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one hydrochloride
J113397 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one Tocris Bioscience
JTE013 Pyrazolopyridine analogue BIOTREND, Tocris Bioscience
JWH133 (3-(1,1-dimethylbutyl)-6,6,9-trimethyl-6a,7,10,10α-tetrahydro-6H-benzo[c]chromene BIOTREND, Sigma-Aldrich, Tocris Bioscience
JYL1421 N-(4-tert-butylbenzyl)-N′-[3-fluoro-4-(methylsulfonylamino)benzyl]thiourea
K31440 Ac-(d-Tyr11,His12,Nle17)sauvagine-(11–40)
Ketanserin 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedione Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
Ki16425 3-(4-[4-{(1-[2-chlorophenyl]ethoxy)carbonylamino}-3-methyl-5-isoxazolyl] benzylsulfanyl) propanoic acid Sigma-Aldrich
KT5720 (9S,10S,12R)-2,3,9,10,11,12-hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1Hdiindolo[1,2,3-fg:3′,2′,1′-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid hexyl ester BIOTREND, Sigma-Aldrich, Tocris Bioscience
L165041 (4-[3-{4-acetyl-3-hydroxy-2-propylphenoxy}propoxyl]phenoxy)acetic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
L655708 11,12,13,13a-tetrahydro-7-methoxy-9-oxo-9H-imidazo[1,5-α]pyrrolo[2,1-c][1,4]benzodiazepine-1-carboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
L689560 trans-2-carboxy-5,7-dichloro-4-phenylaminocarbonylamino-1,2,3,4-tetrahydroquinoline Alexis Biochemicals, Tocris Bioscience
L690330 1-(4-hydroxyphenoxy)ethane-1,1-bisphosphonate Alexis Biochemicals, Tocris Bioscience
L694247 2-[5-[3-(4-methylsulphonylamino)benzyl-1,2,4-oxadiazol-5-yl]-1H-indol-3yl] ethanamine Sigma-Aldrich, Tocris Bioscience
L701324 7-chloro-4-hydroxy-3-(3-phenoxy)phenyl-2(H)quinolone Sigma-Aldrich, Tocris Bioscience
L703606 cis-2(diphenylmethyl)-N-([2-iodophenyl]methyl)-1-azabicyclo[2.2.2]octan-3-amide Alexis Biochemicals, Sigma-Aldrich
L741742 5-(4-chlorophenyl)-4-methyl-3-(1-[2-phenethyl]piperidin-4-yl)isoxazole Tocris Bioscience
L742694 (2(S)-((3,5-bis(trifluoromethyl)benzyl)-oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol-5-yl)methyl)morpholine
L745870 3-[{4-(4-chlorophenyl)piperazin-1-yl}methyl)-1H-pyrrolo[2,3-b]pyridine Sigma-Aldrich, Tocris Bioscience
L750667 iodinated L745870 Sigma-Aldrich
L-AP4 S-2-amino-4-phosphonobutyrate Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
L-CCG-I (2S,3S,4S)α-(carboxycyclopropyl)glycine BIOTREND, Sigma-Aldrich, Tocris Bioscience
LF160687 1-([2,4-dichloro-3-{([2,4-dimethylquinolin-8-yl]oxy)methyl}phenyl]sulfonyl)-N-(3-[{4-(aminoimethyl)phenyl}carbonylamino]propyl)-2(S)-pyrrolidine-carboxamide
LG100268 6-(1-[3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphthalen-2-yl]cyclopropyl)-nicotinic acid
LGD1069 4-(1-[3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-2-naphthyl]ethenyl)-benzoic acid
Linopirdine BIOTREND, Sigma-Aldrich, Tocris Bioscience
LPS Lipopolysaccharide derived from Gram-negative bacteria Alexis Biochemicals, BIOTREND, Sigma-Aldrich
LY278584 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxamide Sigma-Aldrich
LY341495 2S-2-amino-2-(1S,2S-2-carboxycyclopropan-1-yl)-3-(xanth-9-yl)propanoic acid Tocris Bioscience
LY367385 (+)-2-methyl-4-carboxyphenylglycine Tocris Bioscience
LY379268 (—)-2-oxa-4-aminobicylco[3.1.0]hexane-4,6-dicarboxylic acid Tocris Bioscience
LY393675 α-Substituted-cyclobutylglycine
M15 Galanin-(1–13)-substance P-(5–11) amide, also known as galantide Bachem, BIOTREND, Sigma-Aldrich, Cayman
M32 Galanin-(1–13)-neuropeptide Y amide-(25–36) amide Bachem, Sigma-Aldrich
m-3M3FBS 2,4,6-trimethyl-N-(meta-3-trifluoromethylphenyl)-benzenesulfonamide; Calbiochem, Sigma-Aldrich, Tocris Bioscience
MAP4 (S)-2-methyl-2-amino-4-phosphonobutanoate BIOTREND, Sigma-Aldrich, Tocris Bioscience
MBP10 cyclo(6b-410e)(succinyl(6)-d-(2′)Nal7-Arg8-Trp9-Lys10)-NH2
MDL100907 (7)2,3-dimethoxyphenyl-1-[2-(4-piperidine)-methanol]
MDMA 3,4-methylenedioxymethamphetamine Sigma-Aldrich
MEC Mucosa expressed chemokine BIOTREND
Mec Mecamylamine BIOTREND, Sigma-Aldrich, Tocris Bioscience
MEN10627 cyc(2β–5β)(Met-Asp-Trp-Phe-Dap-Leu) BIOTREND, Tocris Bioscience
Methanandamide (R)-(+)-arachidonoyl-1′-hydroxy-2′-propylamide Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
MeTRH pGlu-[Nt-methyl]His-ProNH2 Bachem, Sigma-Aldrich
Mibolerone 7α,17α-dimethyl-1-nortestosterone
Minoxidil 6-(1-Piperidinyl)-2,4-pyrimidinediamine 3-oxide Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
MIP Macrophage inflammatory protein Bachem, BIOTREND, Calbiochem, Sigma-Aldrich
MK886 3-(1-[p-chlorobenzyl]-5-[isopropyl]-3-tert-butylthioindol-2-yl)-2,2-dimethylpropanoic acid methyl ester Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
MK912 (2S,12bS)1′,3′-dimethylspiro(1,3,4,5′,6,6′,7,12b-octahydro-2H-benzo[b]furo[2,3-a]quinolizine)-2,4′-pyrimidin-2′-one Sigma-Aldrich
ML10302 2-(1-piperidinyl)ethyl-4-amino-5-chloro-2-methoxybenzoate Menarini, Sigma-Aldrich
MLA Methyllycaconitine BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
MNQX 6,8-dinitroquinoxaline-2,3,-dione
MPEP 2-methyl-6-(phenylethynyl)-pyridine Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
MPIF-1 Myeloid progenitor inhibitory factor 1
MPP+ 1-methyl-4-phenylpyridinium Sigma-Aldrich
MPPG (RS)α-methyl-4-phosphonophenylglycine Alexis Biochemicals, BIOTREND, Tocris Bioscience
MRS1220 9-chloro-2-(2-furyl)5-phenylacetylamino[1,2,4]triazolo[1,5c]quinazoline Sigma-Aldrich, Tocris Bioscience
MRS1706 N-(4-acetylphenyl)-2-(4-[2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl]phenoxy)acetamide Tocris Bioscience
MRS1754 8-(4-[{(4-cyanophenyl)carbamoylmethyl}oxy]phenyl)-1,3-di(n-propyl)xanthine Sigma-Aldrich, Tocris Bioscience
MRS2179 N6-methyl-2′-deoxyadenosine-3′,5′-bisphosphate Sigma-Aldrich, Tocris Bioscience
MRS2279 2-Chloro-N6-methyl-(N)-methanocarba-2′-deoxyadenosine-3′,5′- bisphosphate Tocris Bioscience
Mus Muscarine Sigma-Aldrich
NADPH Reduced nicotinamide adenosine dinucleotide phosphate Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich
Naltriben BIOTREND, Sigma-Aldrich, Tocris Bioscience
NAPE-PLD N-acylethanolamine-specific phospholipase D
NAS181 (R)-(+)-2-[[[3-(morpholinomethyl)-2H-chromen-8-yl]oxy]methyl] morpholine methane sulphonate BIOTREND, Tocris Bioscience
NBI27914 2-methyl-4-(N-propyl-N-cyclopropanemethylamino)-5-chloro-6-(2,4,6-trichloroanilino)pyrimidine BIOTREND, Sigma-Aldrich, Tocris Bioscience
NBQX 6-nitro-7-sulfamoyl-benz(f)quinoxaline-2,3-dione Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
NBTGR Nitrobenzylthioguanosine Sigma-Aldrich
NBTI Nitrobenzylthioinosine (also known as NBMPR) Sigma-Aldrich
NDGA Nordihydroguiaretic acid BIOTREND, Calbiochem, Sigma-Aldrich
NDP-MSH [Nle4,D-Phe7]α-MSH Bachem, BIOTREND, Calbiochem
NECA Adenosine-5′-N-ethyluronamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
Neuropeptide SF Ser-Leu-Ala-Pro-Gln-Arg-Phe-amide Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
NF023 8,8′-(carbonylbis[imino-3,1-phenylene carbonylimino])bis-1,3,5-naphthalenetrisulphonic acid BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
NFPS N-[3-(4′-fluorophenyl)-3-(4′-phenylphenoxy)propyl]sarcosine BIOTREND, Sigma-Adlrich, Tocris Bioscience
Nic Nicotine Sigma-Aldrich
BNifedipine 1,4-Dihydro-2,6-dimethyl-4-(2-nitrophenyl)-3,5-pyridinedicarboxylic acid dimethyl ester BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
NIL l-N6-(1-iminoethyl)lysine Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
NKH477 6-(3-dimethylaminopropionyl)forskolin hydrochloride Tocris Bioscience
NKY80 2-amino-7-(2-furanyl)-7,8-dihydro-5(6H)-quinazolinone Calbiochem
NMU Neuromedin U BIOTREND, Sigma-Aldrich, Tocris Bioscience
NNC052090 1-(3-[9H-carbazol-9-yl]-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol Tocris Bioscience
NNC711 1-2-([{diphenylmethylene}amino]oxy)ethyl)-1,2,5,6-tetrahydro-3-pyridinecarboxylic acid hydrochloride BIOTREND, Tocris Bioscience
NPC17731 dArg[Hyp3,dHypE(transpropyl)7,Oic8]BK
NS3763 5-carboxyl-2,4-di-benzamido-benzoic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
OAG 1-oleoyl-2-acetyl-sn-glycerol Avanti, Calbiochem, Sigma-Aldrich
ODQ 1H-[1,2,4]oxadiazolo[4,3-a]quinoxalin-1-one Alexis Biochemicals, BIOTREND, Calbiochem, Tocris Bioscience
OHC Hydroxycholesterol Sigma-Aldrich
ONO-AE1-329 16-(3-methoxymethyl)phenyl-ω-tetranor-3,7-dithia-PGE1 Calbiochem
OPC51803 (5R)-2-(1-[2-chloro-4-{1-pyrrolidinyl}benzoyl]-2,3,4,5-tetrahydro-1H-1-benzazepin-5-yl)-N-isopropylacetamide Calbiochem
ORG2058 16α-ethyl-21-hydroxy-19-norpregn-4-ene-3,20-dione
OXE Oxoeicosanoid
Pan Pancuronium BIOTREND, Sigma-Aldrich, Tocris Bioscience
Paz-PC 1-palmitoyl-2-azelaoyl-sn-glycero-3-phosphocholine Alexis Biochemicals, Avanti
PCCG-4 (2S,1′S,2′S,3′R)-2-(2′-carboxy-3′-phenylcyclopropyl)glycine Alexis Biochemicals
PD098059 2-(2-amino-3-methoxyphenyl)-4H-1-benzopyran-4-one Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris
Bioscience
PD102807 9-methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza- BIOTREND, Tocris Bioscience
benzo[a]cyclopenta(h)anthacene-1-carboxylic acid ethyl ester
PD123319 (S)-1-(4-[dimethylamino]-3-methylphenyl)methyl-5-(diphenylacetyl)-4,5,6,7-tetrahydro-1Himidazo[4,5-c]pyridine-6-carboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
PD128907 R-(+)-trans-3,4,4a,10b-tetrahydro-4-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazine-9-ol BIOTREND, Sigma-Aldrich, Tocris Bioscience
PD157672 Boc-(S)Phe-(R)aMePheNH(CH2)7NHCONH2
PD168077 N-methyl-4-(2-cyanophenyl)piperazinyl-3-methylbenzamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
PD184352 2-(2-chloro-4-iodophenylamino)-N-cyclopropylmethoxy-3,4-difluorobenzamide Alexis Biochemicals
PEA 2-phenylethylamine Sigma-Aldrich
Pen5 U-II-4-11 [pencillamine,β,β-dimethylcysteine]5 U-II-4-11
Phenylaceytlrivanil
PIP2 Phosphatidylinositol 4,5-bisphosphate Avanti, BIOTREND, Calbiochem, Roche, Sigma-Aldrich
PIP3 Phosphatidylinositol 3,4,5-trisphosphate Avanti, BIOTREND, Calbiochem
Pirenzepine 5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one dihydrochloride BIOTREND, Sigma-Aldrich, Tocris Bioscience
PIT 2,2′-pyridylisatogen tosylate Tocris Bioscience
PKA Protein kinase A or cyclic AMP-dependent protein kinase BIOTREND, Calbiochem, Sigma-Aldrich
PKC Protein kinase C BIOTREND, Calbiochem, Sigma-Aldrich
PMA Phorbol 12 myristate 13-acetate Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
PMBA 3-[2′-phosphonomethyl[1,1′-biphenyl]-3-yl]alanine Sigma-Aldrich
polyIC Polyinosine-polycytosine Alexis Biochemicals
PPADS Pyridoxalphosphate-6-azophenyl-2′,4′-disulphonate BIOTREND, Sigma-Aldrich, Tocris Bioscience
Ptdlns(3, 4, 5)P3 Phosphatidylinositol (3,4,5)-trisphosphate BIOTREND, Sigma-Aldrich
Pyr3TRH pGlu-His-pyrrolidone
QNB 3-quinuclidinylbenzilate Sigma-Aldrich
R(+)SKF38393 R(+)-7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine Alexis Biochemicals, Sigma-Aldrich, Tocris Bioscience
R(+)SKF81297 R(+)-6-chloro7,8-dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-benzazepine Sigma-Aldrich, Tocris Bioscience
R1881 17β-hydroxy-17α-methyl-estra-4,9,11-triene-3-one, also known as methyltrienolone
R715 AcLys[d Nal7, Ile8][des-Arg9]BK
R848 1-(4-amino-2-ethoxymethyl-imidazo[4,5-c]quinolin-1-yl)-2-methyl-propan-2-ol, also known as resiquimod and S28463
R914 AcLys-Lys-([aMe]Phe5,d-bNal7,Ile8)desArg9BK
RGS2 Regulator of G-protein Signalling 2 (ENSG00000116741)
RJR-2403 (e)-N-methyl-4-(3-pyridinyl)-3-butene-1-amine BIOTREND, Sigma-Aldrich, Tocris Bioscience
Ro154513 methyl-8-azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-α][1,4] benzodiazepine-3-carboxylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
Ro16-6491 N-(2-aminoethyl)-4-chlorobenzamide BIOTREND
Ro201724 4-(3-butoxy-4-methoxyphenyl)methyl-2-imidazolidone Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Ro251553 Ac-His1[Glu8,Lys12,Nle17,Ala19,Asp25,Leu26,Lys27,28,Gly29,30,Thr31]VIP-NH2 (cyclo 21–25)
Ro318220 Bisindoylmaleimidine 1X Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Ro406055 4-([5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl]carboxamido)benzoic acid (also known as AM580) BIOTREND, Tocris Bioscience
Ro415253
Ro600175 (S)-2-(6-chloro-5-fluroindol-1-yl)-1-methyethylamine Tocris Bioscience
RP67580 3αR,7αR-(1-imino-2-[2-methoxyphenyl]ethyl)-7,7-diphenyl-4-perhydroisoindolone BIOTREND, Tocris Bioscience
RS102221 8-[5-(5-amino 2,4-dimethoxyphenyl) 5-oxopentyl]-1,3,8-triazaspiro[4,5]decane-2,4-dione Tocris Bioscience
RS17053 N-[2-(2-cyclopropylmethoxyphenoxy)ethyl]-5-chloro-α,α-dimethyl-1H-indole-3-ethanamide Tocris Bioscience
RS67506 1-(4-amino-5-chloro-2-methoxyphenyl)-3-(1-n-butyl-4-piperidinyl)-1-propanone Tocris Bioscience
RS93520 Z-4-([C3′S,1R,2R,3S,6R]-2C3′-cyclohexyl-3′-hydroxyprop-1-ynyl)-3-hydroxybicyclo(4.2.0)oct-7-ylidene butyrate
RU28318 3-oxo-7-propyl-17-hydroxy-androstan-4-en-17-yl BIOTREND, Tocris Bioscience
RU5135 3a-hydroxy-16-imino-5b-17-azaandrostan-11-one
rutheniumred Ammoniated ruthenium oxychloride Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
RvE1 Resolvin E1 or 5s, 12R, 18R-trihydroxy-6z, 8E, 10E, 14z, 16E-EPA
RX821002 2-(2-methoxy-1,4-benzodioxan-2-yl)-2-imidazoline BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
RY024 Tert-butyl-8-ethynyl-5,6-dihydro-5-methyl-6-oxo-4H-imidazol[1,5-α][1,4]benzodiazepine-,3-carboxylate Tocris Bioscience
Ryanodine 1H-Pyrrole-2-carboxylic acid Alexis Biochemicals, BIOTREND, Calbiochem, Tocris Bioscience
S20098 N-(2-[7-methoxy-1-naphthalenyl]ethyl)acetamide
salicylidene BIOTREND, Tocris Bioscience
salicylhydrazide
SAM S-adenosylmethionine BIOTREND, Sigma-Aldrich
SAM486A 1-guanidinoimino-2,3-dihydroindene-4-carboximidamide, also known as CGP48664
SB200646 N-(1-methyl-5-indonyl)-N'-(3-pyridyl) urea hydrochloride BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB203580 4-(4-fluorophenyl)-2-(4-methylsulphinylphenyl)-5-(4-pyridyl)1H-imidazole Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
SB204070 1-butyl-4-piperidinylmethyl-8-amino-7-chloro-1-4-benzoioxan-5-carboxylate; Sigma-Aldrich
SB204741 N-(1-methyl-5-indoylyl)-N'-(3-methyl-5-isothiazolyl)urea BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB207710 1-butyl-4-piperidinylmethyl-8-amino-7-iodo-1,4-benzodioxan-5-carboxylate
SB224289 1′-methyl-5[[2′-methyl-4′-)5-methyl-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl-2,3,6,7-tetrahydrospiro[furo[2,3-f]indole-3,4′-piperidine]oxalate BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB236057 1′-ethyl-5-(2′-methyl-4′-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carbonyl)-2,3,6,7-tetrahydrospiro[furo[2,3-f]indol3-3,4′-piperidine
SB242084 6-chloro-5-methyl-1-[2-(2-methylpyridyl-3-oxy)-pyrid-5-yl carbamoyl] indoline Sigma-Aldrich, Tocris Bioscience
SB258585 4-iodo-N-[4-methoxy-3-(4-methyl-piperazin-1-yl)-phenyl]-benzenesulphonamide BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB258719 (R)-3,N-dimethyl-N-[1-methyl-3-(4-methylpiperidin-1-yl)propyl]benzene sulphonamide Tocris Bioscience
SB269970 (R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulphonyl)phenol BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB277011 trans-N-(4-[2-{6-cyano-1,2,3,4-tetrahydroisoquinolin-2-yl}ethyl]cyclohexyl)-4-quinolininecarboxamide
SB334867A 1-(2-methyylbenzoxanzol-6-yl)-3-[1,5]naphthyridin-4-yl-urea hydrochloride BIOTREND, Tocris Bioscience
SB366791 N-(3-methoxyphenyl)-4-chlorocinnamide Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
SB408124 (1-(6,8-difluoro-2-methyl-quinolin-4-yl)-3-(4-dimethylamino-phenyl)-urea) BIOTREND, Sigma-Aldrich, Tocris Bioscience
SC19220 1-acetyl-2-(8-chloro-10,11-dihydrobenz[b,f][1,4]oxazepine-10-carbonyl)hydrazine BIOTREND, Sigma-Aldrich, Tocris Bioscience
SC46275 methyl-7-(2β-[6-{1-cyclopenten-1-yl}-4r-hydroxy-4-methyl-1e,5e-hexadienyl]-3α-hydroxy-5-oxo-1R,1a-cyclopentyl)-4Z-heptenoic acid
SC51089 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-[1-oxo-3-(3-pyridinyl)propyl]hydrazide
SC51322 8-Chlorodibenz[b,f][1,4]oxazepine-10(11H)-carboxylic acid, 2-[3-[furanylmethyl)-thio]-1-oxopropyl]hydrazide
SC560 5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-trifluoromethylpyrazole Alexis Biochemicals, Calbiochem, Sigma-Aldrich, Tocris Bioscience
SCH23390 7-chloro-8-hydroxy-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine BIOTREND, Sigma-Aldrich, Tocris Bioscience
SCH90511 (+)-(2S)-5,5-dimethyl-2-morpholineacetic acid Tocris Bioscience
S-ENBA (2S)-N6-(2-endonorbanyl)adenosine Sigma-Aldrich, Tocris Bioscience
SEW2871 5-(4-phenyl-5-trifluoromethylthiophen-2-yl)-3-(3-trifluoromethylphenyl)-(1,2,4)-oxadiazole BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
SIB1757 6-methyl-2-(phenylazo)-3-pyrindol BIOTREND, Sigma-Aldrich, Tocris Bioscience
SIB1893 ([phenylazo]-3-pyrindole)-2-methyl-6-(2-phenylethenyl)pyridine Alexis Biochemicals, BIOTREND, Sigma-Aldrich, Tocris Bioscience
SKF83566 (−)-7-bromo-8-hydroxy-3-methyl-1-phenyl-2,3,4,5-tetrahydro-3-benzazepine BIOTREND, Sigma-Aldrich, Tocris Bioscience
SKF89976A 1-(4,4-diphenyl-3-butenyl)-3-piperidinecarboxylic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
SKF96265 1-(β-(3-(4-methoxyphenyl)propoxy)-4-methoxyphenethyl)-1H-imidazole hydrochloride BIOTREND, Calbiochem
SLC Secondary lymphoid tissue chemokine Sigma-Aldrich
SQ27986 [1S-[1B,2B(5Z),3A(1E, 3S)4B]]7-[3-(3-cyclohexyl-3-hydroxy-1-propenyl)-7-oxabicyclo[2.2.1]hept-2-y]5-heptenoic acid
SR142801 (s)-(N)-(1-[3-{1-benzoyl-3-(3,4-dichlorophenyl)piperidin-3-yl}propyl]-4-phenylpiperidin-4-yl)-N-methylacetamide
SR142948A 2-([5-{2,6-dimethoxyphenyl}-1-{4-(N-[3-dimethylaminopropyl]-N-methylcarbamoyl)-2-isopropylphenyl}-1H-pyrazole-3-carbonyl]amino)adamantane-2-carboxylic acid hydrochloride Tocris Bioscience
SR2640 2-(3-[2-quinolylmethoxy]phenylamino)benzoic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
SR48968 (S)-N-methyl-N-(4-acetylamino-4-phenylpiperidino)-2-(3,4-dichlorophenyl)butylbenzamide, also known as saredutant Sigma-Aldrich
SR57227 4-amino-(6-chloro-2-pyridyl)-1-piperidine hydrochloride BIOTREND, Sigma-Aldrich, Tocris Bioscience
SR95531 2-(3′-carboxy-2′-propyl)-3-amino-6-p-methoxyphenylpyridazinium bromide BIOTREND, Sigma-Aldrich, Tocris Bioscience
SRA125543A 4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1S)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]5-methyl-N-(2-propynyl)-1,3-thiazol-2-amine hydrochloride
SSR126768A 4-chloro-3-[(3R)-(+)-5-chloro-1-(2,4-dimethoxybenzyl)-3-methyl-2-oxo-2,3- dihydro-1H-indol-3-yl]-N-ethyl-N-(3-pyridylmethyl)-benzamide,hydrochloride
Str Strychnine Sigma-Aldrich, Tocris Bioscience
Suramin Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
Sux Succinylcholine BIOTREND, Calbiochem, Sigma-Aldrich
T0070907 2-chloro-5-nitro-N-(4-pyridyl)benzamide BIOTREND, Tocris Bioscience
T226296 (–)-N-[6-(dimethylamino)-methyl]-5,6,7,8-tetrahydro-2-naphthalenyl]-4′-fluoro[1,1′-biphenyl]-4-carboxamide
TARC T-cell and activation-related chemokine Bachem, BIOTREND, Sigma-Aldrich
TBPS Tert-butylbicyclophosphorothionate Sigma-Aldrich
TEA Tetraethylammonium BIOTREND, Calbiochem, Sigma-Aldrich
THIQ N-([3R]-1,2,3,4-tetrahydroisoquinolinium-3-ylcarbonyl)-(1R)-1-(4-chlorobenzyl)-2-(4-cyclohexyl-4-[1H-1,2,4-triazol-1ylmethyl]piperidin-1-yl)-2-oxoethylamine
TIPP Tyr-Tic-Phe-Phe Bachem, Sigma-Aldrich
TMB-8 8-(diethylamine)octyl-3,4,5-trimethoxybenzoate BIOTREND, Calbiochem, Sigma-Aldrich
TNP-ATP 2′,3′-O-(2,4,6-trinitrophenyl)adenosine 5′-triphosphate Sigma-Aldrich, Tocris Bioscience
TPMPA (1,2,5,6-tetrahydropyridine-4-yl)methylphosphinic acid BIOTREND, Sigma-Aldrich, Tocris Bioscience
TTNPB (E)-4-(2-[5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl]-1-propenyl)benzoic acid BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
tyrphostin AG1478 N-(3-chlorophenyl)-6,7-dimethoxyquinazolin-4-amine hydrochloride Alexis Biochemicals, Sigma-Aldrich, Tocris Bioscience
tyrphostin AG879 α-cyano-(3,5-di-t-butyl-4-hydroxy)thiocinnamide Alexis Biochemicals, Calbiochem, Sigma-Aldrich, Tocris Bioscience
U0126 1,4-diamino-2,3-dicyano-1,4-bis(o-aminophenylmercapto)butadiene Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
U46619 11α,9α-epoxymethano-PGH2 Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
U69593 5a,7a,8b-(–)-N-methyl-N-(7-[1-pyrrolidinyl]-1-oxasipro(4,5)dec-8-yl)benzene acetamide Alexis Biochemicals, Sigma-Aldrich
U73122 1-(6-[{(17β)-3-methoxyestra-1,3,5[10]-trien-17-yl}amino]hexyl)-1H-pyrrole-2,5-dione Alexis Biochemicals, BIOTREND, Calbiochem, Tocris Bioscience
U75302 6-(6-(3-hydroxy-1E,5Z-undecadien-1-yl)-2-pyridinyl)-1,5-hexanediol
UBP296 (RS)-3-2-carboxybenzyl)willardiine BIOTREND, Tocris Bioscience
UH301 5-fluoro-8-hydroxy-2-(dipropylamino) tetralin Sigma-Aldrich
UK14304 5-bromo-6-[2-imidazolin-2-ylamino]quinoxaline BIOTREND, Sigma-Aldrich, Tocris Bioscience
Val2TRH pGlu-Val-ProNH2
WAY100635 N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridyl)-cyclohexanecarboxamide trichloride Sigma-Aldrich
WAY-855 3-amino-tricyclo[2.2.1.02.6]heptane-1,3-dicarboxylic acid
WIN35428 2β-carboxymethy-3β-(4-fluorophenyl)tropane Sigma-Aldrich
WIN55212-2 (R)-(+)-[2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo-[1,2,3-de]-1,4-benzoxazin-6-yl]-1-Naphthalenylmethanone mesylate BIOTREND, Sigma-Aldrich, Tocris Bioscience
WY14643 N-(3-[2-quinolinylmethoxy]phenyl)-trifluoromethanesulphonamide Alexis Biochemicals, BIOTREND, Calbiochem, Sigma-Aldrich, Tocris Bioscience
XAC 8-(4-[{([{2-aminoethyl}amino]carbonyl)methyl}oxy]phenyl)-1,3-dipropylxanthine, also known as xanthine amine congener Sigma-Aldrich
XE991 10,10-bis(4-pyridinylmethyl)-9(10H)-anthracene BIOTREND, Tocris Bioscience
xestospongin C Calbiochem, Sigma-Aldrich
YC-1 3-(5′-hydroxymethyl-2′-furyl)-1-benzylindazole Alexis Biochemicals, Calbiochem, Sigma-Aldrich
BZD7288 4-(N-ethyl-N-phenyl-amino)-1,2-dimethyl-6-(methylamino)pyrimidinium chloride BIOTREND, Tocris Bioscience
ZM241385 4-(2-[7-amino-2-{2-furyl}{1,2,4}triazolo{2,3-a}{1,3,5}triazin-5-ylamino]ethyl)phenol BIOTREND, Calbiochem, Tocris Bioscience
α-Dendrotoxin Bachem, BIOTREND, Sigma-Aldrich
α-Methyl-5-HT α-Methyl-5-hydroxytryptamine BIOTREND, Tocris Bioscience
αβ-MeATP αβ-Methylene-adenosine 5′-triphosphate Sigma-Aldrich
βγ-MeATP βγ-Methylene-adenosine 5′-triphosphate Sigma-Aldrich
µ-Conotoxin GIIIA Bachem
ω-Agatoxin IVA Alexis Biochemicals, Bachem, BIOTREND, Sigma-Aldrich
ω-Conotoxin GVIA Alexis Biochemicals, Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience
ω-Conotoxin MVIIC Alexis Biochemicals, Bachem, BIOTREND, Sigma-Aldrich, Tocris Bioscience

Articles from British Journal of Pharmacology are provided here courtesy of The British Pharmacological Society

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