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Aqueous oxidative Heck reactions with protein-bound alkenes according to Scheme 1 monitored by LC-MS
| R1 | R2 | R3 | Catalyst/boronic acid | Conversion |
|---|---|---|---|---|
| H |  |
50:300 | full | |
| H |  |
20:100 | full | |
| H |  |
10:50 | ≈85 % | |
 |
4-OMe |  |
20:100 | full |
| 4-OT R61C-1 | ||||
| 4-COOMe |  |
20:100 | ≈85 % | |
| 3-NH-dansyl |  |
20:100 | full | |
 |
H |  |
20:100 | ≈70 % |
| 4-OT R61C-2 | ||||
 |
H |  |
20:100 | ≈5 % |
| 4-OT R61C-3 | ||||
 |
H |  |
20:100 | no |
| 4-OT R61C-4 |
