Table 2. TAM and 1-HP Binding to SULT1A1.
ligand | SULT1A1 species | Kd (μM)a |
---|---|---|
TAM | E | 0.67 (0.08) |
TAM | E·(PAP)2 | 0.65 (0.07) |
TAM | E·PAP | 13 (2) |
1-HP | E | 8 (0.5) |
1-HP | E·(PAP)2 | 0.025 (0.001) |
1-HP | E·PAP | 0.025 (0.0010) |
Values in parentheses indicate one standard deviation.