Table 1. Comparison of selected Stat5a/b inhibitors in efficacy of inhibition of Stat5a/b tyrosine phosphorylation (pYStat5a/b), as detected by Western blot analysis.
Publication (Fig. of Interest): | Inhibitor Name: | pYStat5a/b Inhibition (µM): |
Nam et al. 2012 (Fig. 2A) | E804 | 10-20 |
Nelson et al. 2011 (Fig. 2A) | Pimozide | >10 |
Elumalai et al. 2015 (Fig. 4C) | Stafib-1 (Comp. #17) | 10 |
Müller et al. 2008 (Fig. 3A) | Comp. #6 | 400 |
Page et al. 2012 (Fig. 2A) | BP-1-107 BP-1-108 SF-1-087 SF-1-088 |
40 |
Cumaraswamy et al. 2014 (Fig. 4A) | AC-3-019 | 15 |
Liao et al. 2015 (Fig. 2F) | IST5-002 | 5 |