Table 1.

Summary of the biological activities of synthetic CDXs inspired in natural xanthones.

CDXs	Biological Activities	Ref.
Kielcorin derivatives 2–9	Antitumor and protein kinase C inhibition	[56,58,59,61]
Psorospermin derivatives 11–15	Antitumor	[64]
Muchimangin derivatives 16–20	Antimicrobial	[66]
Mangiferin derivatives 21–57	Antipyretic, antimicrobial, analgesic, antioxidant, anti-inflammatory, antidiabetic, anticoagulant and antiplatelet	[68,72,73,75,76,77,78,81,82,83,86]
α-Mangostin derivatives 58–70	Antimicrobial, hemolytic and antimycobacterial	[91,95,96,97,98,99,118]
Caged xanthones 71–155	Antimalarial, antitumor, anti-proliferation and anti-angiogenesis	[106,108,109,111,113,114,115,116,117,119,120]